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Benzodiazepines (view source)

Revision as of 15:35, 3 March 2009

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→‎Benzodiazepine Antagonists

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==Benzodiazepine Antagonists==

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Benzodiazepine antagonists have no intrinsic efficacy, but prevent agonist interaction with receptors. Examples include flumazenil, which is used in man following benzodiazepine overdose.

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==Inverse Agonists==

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Inverse agonists act at the GABA receptor to close Cl<sup>-</sup> channels. They promote convulsions.

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